For medisinbytte ved institusjoner henvises til §7 i Forskrift om legemiddelhåndtering for virksomheter og helsepersonell som yter helsehjelp
Normally, acetaminophen is used for the remedy of gentle to moderate ache and reduction of fever. It is on the market above the counter in several kinds, the most common being oral varieties.
Legemiddel mot psykoser. I psykiatrien brukes benevnelsen antipsykotika synonymt med nevroleptika eller psykoleptika.
Et syndrom som kjennetegnes av svikt i det CNS i forbindelse med leversvikt. Symptomer er blant annet fatigue og forvirring som ofte forverres til koma, tremor i hender og øye- og muskelrykninger.
Ammende skal ikke bruke kodeinholdige preparater sammenhengende utover two–three dager. Diebarn bør observeres med tanke på slapphet og sedasjon. Kvinner med ultrarask genotype av CYP2D6 vil i høy grad kunne omdanne kodein til morfin.
The proportion of the systemically absorbed rectal dose of acetaminophen is inconsistent, demonstrated by major dissimilarities while in the bioavailability of acetaminophen following a dose administered rectally.
Substans som hemmer virkningen av en annen substans ved konkurrerende binding til reseptorer. Reseptorer finnes bl.
Nevertheless acetylsalicylic acid (aspirin) is surely an irreversible inhibitor of COX and right blocks the Energetic web-site of the enzyme, studies have revealed that acetaminophen (paracetamol) blocks COX indirectly. Studies also suggest that acetaminophen selectively blocks a variant type of the COX enzyme that is unique from your recognized variants COX-one and COX-2. This enzyme is known as COX-three
Sykelig forandring av leveren der det dannes bindevev i stedet for leverceller, slik at leverfunksjonen ødelegges.
Overdose and liver toxicity Acetaminophen overdose could possibly be manifested by renal tubular necrosis, hypoglycemic coma, and thrombocytopenia. From time to time, liver necrosis can come about as well as liver failure.
is indicated for that management of moderate to moderate discomfort, the administration of average to extreme pain with adjunctive opioid analgesics, along with the reduction of fever.
Ingen mistanke om fosterskadelig effekt ved ordinary dosering. Ved intoksikasjoner er det høy frekvens av fosterdød og spontanaborter
Induksjon av metabolismen av paracetamol i lever, både til inaktive metabolitter og til den levertoksiske metabolitten NAPQI.
Acetaminophen is definitely an analgesic more info drug utilized by itself or in combination with opioids for discomfort administration, and being an antipyretic agent.
Animal and clinical experiments have established that acetaminophen has both equally antipyretic and analgesic consequences. This drug has long been shown to lack anti-inflammatory effects. As opposed to the salicylate drug course, acetaminophen does not disrupt tubular secretion of uric acid and would not affect acid-foundation harmony if taken for the advisable doses.
Due to its lower possibility of producing allergic reactions, this drug may be administered in individuals who are intolerant to salicylates and people with allergic tendencies, which include bronchial asthmatics. Distinct dosing suggestions needs to be adopted when administering acetaminophen to little ones.